The IUPHAR/BPS Guide to PHARMACOLOGY complete ligand list

Low molecular weight, non-polymeric compounds produced via either total synthesis or semi-synthetic processes.

A  B  C  D  E  F  G  H  I  J  K  L  M  N  O  P  Q  R  S  T  U  V  W  X  Y  Z 

Ligand name ID Synonyms
A Back to top
852A 9025
A1120 8792 A 1120, compound 33 [PMID: 24835984]
A-119637 490 A 119637, A119637
A-123189 491 A 123189, A123189
A134974 5130 A 134974, A-134974
A192621 1009 A 192621, A-192621
A-196 8949
A286982 6592 A 286982, A-286982
A-304121 1258 A 304121, A304121
A317491 4115 A 317491, A-317491
A-317567 4116 A 317567, A317567
A-317920 1216 A 317920, A317920
A331440 4023 A 331440, A-331440
A-349821 1217 A 349821, A-349,821, A349821
A-366 8238 A 366, A366
A-381393 8441 A 381393, A-381,393
A412997 3301 A-412,997, A-412997
A425619 4117 A 425619, A-425619
A438079 4118 A 438079, A-438079
A-443654 8204 A 443654, A443654
A-582941 3995 A 582941, A582941
A61603 480 A 61603, A-61603
A-674563 5655 A 674563, A674563
A68930 6077 A 68930, A 70108, A 70360, A-68930, A-70108, A-70360, A70108, A70360
A740003 4119 A 740003, A-740003
A778317 4120 A 778317, A-778317
A-794278 6354 A 794278, A794278, compound 1ac [PMID: 16279797]
A-794282 6211 A 794282, A794282, compound 1n [PMID: 16279797]
A-803467 5734 A 803467, A803467
A804598 4121 A 804598, A-804598
A839977 4122 A 839977, A-839977
A-841720 3953 A 841720, A841720
A-850002 6355 A 850002, A850002, compound 28b [PMID: 16279797]
A-85380 5460 A 85380, A85380
A-867744 3986 A 867744, A867744
A-935142 7661 A 935142, A935142
A-967079 6280 A 967079, A967079
[3H]A317491 5407 [3H]A 317491, [3H]A-317491
[3H]A-585539 3974
[3H]A778317 4076
[3H]A804598 5408 [3H]A 804598
[3H]A81988 3938 [3H]-A81988
AAE-M-PBP-amine 8289 acetylaminoethyl-methyl-phenylbutoxyphenyl-amine
Abbott 14c 5871 2,4-diaminopyrimidine-based antagonist, 14c
ABC294640 6624 ABC 294640, ABC-294640
abediterol 9326 LAS-100977
abemaciclib 7382 CS-1230, HY-16297A, LY 2835219, LY2835219
abexinostat 8366 CRA-024781, PCI-24781
abiraterone 6745
abiraterone acetate 9288 Zytiga
ABL127 8608 ABL 127, ABL-127
AB-MECA 416
[125I]AB-MECA 436 [125I]-AB-MECA, [125I]5-[6-[(4-aminophenyl)methylamino]purin-9-yl]-3,4-dihydroxy-N-methyl-oxolane-2-carboxamide, [125I]N(6)-(4-amino-3-iodobenzyl)adenosine-5'-N-methyluronamide
AB-NECA 434 aminobenzyl-5'-N-ethylcarboxamidoadenosine
abnormal cannabidiol 5526 Abn-CBD, CAY10429
[125I]ABOPX 452 [125I]3-(3,4-aminobenzyl)-8-(4-oxyacetate)phenyl-1-propyl-xanthine
ABT-239 1218 ABT 239, ABT239
ABT-288 6927 ABT 288, ABT288
ABT-299 1849 ABT 299, ABT299
ABT-384 7357 ABT 384, ABT384
ABT-491 1850 ABT 491, ABT491
ABT-639 7721 ABT 639, ABT639
ABT-670 8439 ABT 670, ABT670, compound 6b [PMID 17149874]
ABT702 5131 ABT 702, ABT-702
ABT-737 8320 ABT 737, ABT737, compound 2 [PMID 17256834]
AC-186 8897 AC 186
AC-260584 334 AC 260584, AC260584
AC261066 4054 AC 261066, AC-261066
AC262620 4017 AC 262620, AC-262620
AC262970 4018 AC 262970, AC-262970
AC263093 4020 AC 263093, AC-263093
AC265347 3947 AC 265347, AC-265347
AC-42 289 AC 42, AC42
AC430 9177 AC-430
AC45594 5422 4-(heptyloxy)benzolol, 4-heptoxyphenol
AC55649 4055 AC 55649, AC-55649
AC710 8095 AC 710, AC-710
AC-7954 2151 AC 7954, AC7954
AC-90179 174 AC 90179, AC90179
ACAA 2443 ACA
acadesine 5133 AICA-riboside, AR-100, SCH-900395
acalabrutinib 8912 ACP-196, Example 6 [US20140155385 A1]
acamprosate 7106 Campral®
acarbose 6791 BAY-G 5421, BAY-G-5421, Glucobay®, Precose®
Ac-DEVD-CHO 6527
ACDPP 3388
acebutolol 7107 IL-17803A, Sectral®
(-)-aceclidine 288 R-(-)-aceclidine
(+)-aceclidine 286 S-(+)-aceclidine
acelarin 7389 NUC-1031
acenocoumarol 9015 Sinthrome®, Sintrom®
ACET 4123
acetamide 4661 ethanamide, methylformamide
acetazolamide 6792 Diamox®
acetoacetic acid 4522 acetoacetate, diacetic acid
acetohexamide 6793 Dymelor®
1'-acetoxychavicol acetate 6298
[3H]acetylcholine 8593
acetyldigitoxin 6794 acetyldiginatin, Acylanid®, alpha-acetyldigitoxin
acetyl-podocarpic dimer 2753 APD, acetyl podocarpic acid anhydride
aciclovir 4829 acyclovir, Zovirax®
acifran 1595 AY-25712, D02753, reductol
acipimox 1596 Olbetam®
acitretin 7598 Ro-101670000, Soriatane®
aclidinium 7449 LAS W-330, LAS-34273, Tudorza Pressair®
[35S]ACPPB 4584 [35S]-ACPPB
ACPT-I 1408 1-aminocyclopentane-1,3,4-tricarboxylic acid
acrolein 2418
acrylamide 4553
4-acryloylphenol 8841 compound 6
ACT-335827 9122 ACT 335827, compound 9 [PMID: 23589487]
ACT-462206 9303 compound 24 [PMID: 25147058]
acumapimod 9203 BCT 197, BCT-197, BCT197, compound A [WO2013139809]
Ac-VEID-CHO 8566 acetyl-Val-Ile-Asp-aldehyde
ACY-241 9426 citarinostat (proposed INN), HDAC-IN-2
AD-5061 2663 AD 5061, AD 7057, AD-7057, AD5061, AD7057
AD5075 2701 AD 5075, AD-5075
[3H]AD5075 2702 [3H]-AD5075
adapalene 5429 Differin®
adenophostin A 4124
ADL5747 9003 ADL 5747, ADL-5747, compound 36 [PMID: 19694468]
ADL5859 9004 ADL 5859, ADL-5859, compound 20 [PMID: 18788723]
[35S]ADPβS 3408
(+)-ADTN 932 (+)-ADTN (aminotetralin-6,7-diol)
ADX-47273 1420 ADX 47273, ADX47273
ADX71743 6217 ADX 71743, ADX-71743
ADX88178 6238 ADX 88178, ADX-88178
AE9C90CB 8586
AEE788 7643 AEE 788, NVP-AEE788
AF353 4125 AF 353, AF-353
afatinib 5667 BIBW2992, Gilotrif®
AFD(R) 2937
AFDX384 3264 AF-DX 384, AFDX-384
[3H]AF DX-384 368 [3H]AF-DX 384
afegostat 7410 IFM, iso-fagomine, isofagomine
AFP-07 1962 AFP 07, AFP07
afuresertib 7890 GSK 2110183, GSK-2110183, GSK2110183
AG-09/1 5833 AG-09/1 [benzimidazole derivative], ST024252
AG 1024 5912 AG-1024, AG1024, tyrphostin AG 1024
AG-11/03 5832 AG-11/03 [benzimidazole derivative], STK220090
AG 112 5913 AG-112, AG112, tyrphostin A48, tyrphostin AG 112
AG 1295 5914 AG-1295, AG1295
AG 1296 5915 AG-1296, AG1296, tyrphostin AG-1296
AG-14 5835 AG 14, AG14
AG14361 8094 AG 14361, AG-14361
AG1478 4862 AG 1478, AG-1478, tyrphostin AG1478
AG-26 6268 AG 26, AG26
AG 490 5916 AG-490, tyrphostin AG490, tyrphostin B42
AG879 4863 AG 879, AG-879, tyrphostin AG879
AG 9 5917 AG-9, AG9, tyrphostin 1, tyrphostin A1
AGI-5198 9240
AGK2 8099 AGK 2, AGK-2
AGL 2043 5918 AGL-2043, AGL2043, HMS3229A05
AGN 191976 6071 AGN-191976, AGN191976
AGN192093 3387 AGN 192093, AGN-192093
AGN193109 2640 AGN 193109, AGN-93109
AGN193836 2649 AGN 193836, AGN-193836
AGN194204 2811 AGN 194204, AGN-194204
AGN 211334 5455 AGN-211334, AGN211334
agomelatine 198 S20098, Thymanax®, Valdoxan®
AG-041R 901 AG 041R, AG041R, LS-83786
AH 11110 8461 AH-11110, AH11110
AH13205 1928 AH 13205, AH-13205
AH23848 1949 (-)-AH23848, (-)AH23848, AH 23848, AH-23848
AH6809 1896 AH 6809, AH-6809
(S)-4-AHCP 4069
AHPN 3431 CD 437, CD437, Ro 47-2077
AH23848 (racemic) 1950 AH 23848, AH-23848
AIDA 1376 GNF-Pf-1401, UPF 523, UPF523
(+)-AJ76 970
AK198 8637
AKK(thioAc)LM21 8816
AKN-028 7969 AKN 028, AKN028
Akt inhibitor IV 5919 GNF-PF-254
Akt inhibitor VIII 5921 isozyme-selective, Akti-1/2
Akt inhibitor X 5922 10-DEBC, NCGC00167772-01
AL12180 3386 5,6-dihydro-4,5-didehydro-11-deoxy-11-oxa-16-(3-chlorophenoxy)-ω-tetranor-PGF2α, AL-12180
AL-8810 1956 AL 8810, AL8810
AL-37350A 160 AL 37350A, AL37350A
Ala(1-naph)-Pro-CN 8607
alcaftadine 7587 Lastacaft®, R-89674
alectinib 7739 AF802, Alecensa®, CH5424802
aleglitazar 7405 R-1439, Ro-0728804
alemcinal 1444 ABT 229, ABT-229, ABT229
alendronate 3141 ABDP, BPH 1, Fosamax®, MK-217
Alexa-488-telenzepine 8600
alfentanil 7108 Alfenta®, R-39209, Rapifen®
alfuzosin 7109 SL-77499-10, SL-7749910, Uroxatral®
alimemazine 7237 Nedeltran®, trimeprazine
alisertib 7790 MLN-8237
aliskiren 4812 CGP-060536B, SPP100, Tekturna®
alkylbenzene sulfonate 2362
alkyl glycerol phosphate 18:1 6994 AGP 18.1
alkyl OMPT 2913
allopurinol 6795 Aloprim®, BW-56-158, BW-56158, Zyloprim®
alloswitch-1 8543 trans-alloswitch-1
alloxazine 456 alloxazin, isoalloxazine
all-trans-4-oxo-retinoic acid 2741 4-oxoretinoic acid, Ro 12-4824
1-allyl-2-[3-(isopropylamino)propoxy]-9H-carbazole 3136
1-allyl-2-[3-(isopropylamino)propoxy]-9H-xanthen-9-one 3135
allyl isothiocyanate 2420
almorexant 2886 ACT-078573
almotriptan 7110 Axert®, LAS-31416, PNU-180638E
alniditan 120 R-91274
[3H]alniditan 117 R-91274
alogliptin 6319 Nesina®, SYR-322, Vipidia®
aloisine 5923 IN1538, RP106
aloisine A 5924 RP107
alosetron 2296 GR68755, Lotronex®
alpelisib 7955 BYL 719, BYL-719, NVP-BYL719
alpha-ketothiazole analogue 36 6549
alpha-methyltyrosine 6956 Demser®, metyrosine, MK-781
alphaxalone 5461 5α-alphaxalone, alfadione, alfaxalone, GR 2/234
alprazolam 7111 Niravam®, U-31889, Xanax®
alprenolol 563 Atenenol®
ALRT 1550 2740
alsterpaullone 5925 9-nitropaullone, NSC-705701
alsterpaullone 2-cyanoethyl 5926 alsterpaullone derivative7
[18F]altanserin 3242 [18F]altanserin (PET ligand)
altiratinib 9174 DCC-270, DCC-2701, DP-5164
altretamine 7112 Hexalen®
alvelestat 6476 AZD 9668, AZD-9668, AZD9668, KB-105160
alvimopan 7471 ADL 8-2698, Entereg®
alvocidib 5680 flavopiridol, HL 275, HMR 1275, L 86-8275, L 868275, MDL-107826A, NSC-649890
ALX 1393 4622 ALX-1393, ALX1393, O-[2-benzyloxyphenyl-3-flurophenyl]methyl-L-serine
ALX 1405 4767 ALX-1405, ALX1405
AM095 6988 AM 095, AM-095
AM1241 3316 AM 1241, AM-1241
AM251 3317 AM 251, AM-251
AM281 741 AM 281, AM-281
AM-630 750 6-iodopravadoline, AM 630, AM630
AM6538 9338 4-(4-(1-(2,4-dichlorophenyl)-4-methyl-3-(piperidin-1-ylcarbamoyl)-1 H-pyrazol-5- yl)phenyl)but-3-ynyl nitrate, compound 10 [WO2010104488], Example 2 [WO2010104488]
AM7 8292 AM 7, AM-7, pyrimidone, 22
AM7499 9257 compound 3b [PMID: 27367336]
AM966 2905 AM 966, AM-966
[123I]AM251 744
AMA 5134 S-(5'-deoxy-5'-adenosyl)-methylthioethyl-hydroxylamine
amantidine 4128 Symadine®
4-AMBA 4702
ambrisentan 3951 Letairis®
amcinonide 7060 CL-34699, Cyclocort®
AMD070 8580 AMD 070, AMD-070, compound 2 [PMID: 20297846]
amelubant 8463 BIIL 284, BIIL-284
amesergide 199 LY-237733, LY237733
amfenac 7565 AHR-5850D, Fenazox® (Japan)
amg-1 8227
AMG319 8917 AMG 319, AMG-319
AMG-337 8913 compound 24 [PMID: 19819693]
AMG517 4129 AMG 517, AMG-517
AMG628 4130 AMG 628, AMG-628
AMG7703 5803 AMG 7703, AMG-7703
AMG-837 6485 AMG 837, AMG837
AMG-900 8060 AMG 900, AMG900
AMG 9810 6347 AMG-9810, AMG9810
AMI-1 7028 AMI 1, AMI1
amibegron 568 SR 58611, SR-58,611A, SR-58611A, SR58611A
amidephrine 514
amifampridine 8032 3,4-DAP, 3,4-diaminopyridine, Firdapse®, Zenas®
amiloride 2421 amiloride HCl, Midamor®
aminobenzovesamicol 4768 compound 11 [PMID: :7702637], M-iodobenzyltrozamicol
2(S)-amino-6-boronohexanoic acid 5107 ABH
6-aminocaproic acid 6574 ε-aminocaproic acid, Amicar®, EACA
aminoethoxyvinylglycine 8860 AVG, aviglycine
aminoglutethimide 7054 Cytadren®
2-amino-4-methylpyridine 5111
aminopurvalanol A 5927 NG-97
5-aminosalicylate 4655 5-ASA, 5-aminosalicylic acid, mesalamine
2-amino-3-sulfinopropanoic acid 4695 3-sulfinoalanine, cysteine sulfinate
2-amino-uridine-5'-monophosphate 6201 compound 13g [PMID: 21417463], iso-CMP
amiodarone 2566 amiodarone hydrochloride, Cordarone®
amiselimod 9319 Example 1 [US20090137530], MT-1303, MT1303
amisulpride 963 (±)-amisulpride
amitriptyline 200 amitryptiline, Elavil®, Endep®
amlexanox 7113 AA-673, Amlexanox®, Aphthasol®, CHX-3673
amlodipine 6981 amlodipine besylate, amlodipine maleate, Norvasc®, UK-4834011
ammonium carbonate 4509
AMMTC 3385
AMN082 1441 AMN 082, AMN-082
amoxapine 201 amoxipine, Asendin®
AMPA 4131
[3H]AMPA 4077
amphetamine 4804 (±)-amphetamine, Amphetamine Sulfate®, DL-amphetamine
AMTB 4132
amthamine 4025
amuvatinib 7932 MP 470, MP-470, MP470
anacetrapib 8400 MK-0859
anagrelide 7114 Agrylin®, BL-4162a, Xagrid®
analog 3 [Vlattas et al., 1996] 7994
anastrozole 5137 Arimidex®
anatibant 679 LF 16-0687, LF160687
ancriviroc 804 SCH 351125, SCH-351125, SCH-C
[3H]ancriviroc 802 [3H]SCH 351125, [3H]Sch-351125
andarine 7849 GTX-007, GTX007
androstanol 2760 5α-androstan-3α-ol
4,9-anhydro-tetrodotoxin 5730 4,9-ah-TTX, 4,9-anhydro-TTX
anileridine 7115 Leritine®
aniracetam 4133
anisindione 6960 Miradon®
antalarmin 3489
ANTAQ 8671 compound 5
antazoline 7116
9-anthroic acid 4113 9-AC, anthracene-10-carboxylic acid
anti-BrP-LPA 6987
A1P 8806 compound 10 [PMID: 20441173]
AP18 4134 AP 18, AP-18
[3H]AP4 1412
Ap3a 5454 diadenosine triphosphate
Ap5a 5453 diadenosine pentaphosphate
APA 5139 1-aminooxy-3-aminopropane
apadenoson 3290 ATL-146e, BMS-068645
apafant 1860 WEB 2086 BS, WEB-2086
[3H]apafant 1859 [3H]WEB 2086
apalutamide 9043 ARN-509, ARN509, JNJ-56021927
apatinib 7648 YN968D1
2-APB 2433 2-aminoethoxydiphenyl borate, 2-aminoethoxydiphenylborane
apitolisib 7888 GDC-0980, GDC0980, RG-7422, RG7422
apixaban 6390 BMS-562247, Eliquis®
aplaviroc 805 AK-602, GW 873140, GW873140A
3-APMPA 1080 CGP 35024, CGP35024, SK&F 97541, SKF 97541, SKF-97,541
APNEA 417 N6-2-(4-aminophenyl)ethyladenosine
[125I]APNEA 462 [3H]N6-2-(4-aminophenyl)ethyladenosine
apomorphine 33 Apokyn®, Ixense®, Uprima®
3-APPA 1081 3-aminopropanephosphinic acid, APPA, CGP-27492
4-APPES